From: Do polyphenols enter the brain and does it matter? Some theoretical and practical considerations
PP | Test conc. (μM) | Incubation time | Cell line | Intracellular conc. | Study |
---|---|---|---|---|---|
Apigenin | 50 | 2Â h | Caco-2 | ~1.2Â nmol/mg protein | Yokomizo and Moriwaki (2006)a |
Kaempferol | ~1.8Â nmol/mg protein | ||||
Luteolin | ~1.3Â nmol/mg protein | ||||
Quercetin | ~0.9Â nmol/mg protein | ||||
Myricetin | ND | ||||
Myricetrin | ND | ||||
Rutin | ND | ||||
Isoquercitrin | ND | ||||
Quercetin | 500 | 1Â h | H4IIE | 33.4Â nmol/106 cells | Watjen et al. (2005) |
Fisetin | 12.67Â nmol/106 cells | ||||
Myricetin | 0.22Â nmol/106 cells | ||||
Morin | 2.35Â nmol/106 cells | ||||
Taxifolin | 0.2Â nmol/106 cells | ||||
Rutin | 0 | ||||
Catechin | 0 | ||||
EC | 50 | 1Â h | Caco-2 | 0 | Vaidyanathan and Walle (2003)a |
(+)-Catechin | ~150Â pmol/mg protein | ||||
ECG | ~3,000Â pmol/mg protein | ||||
EGCG | ~2,400Â pmol/mg protein | ||||
Quercetin | 5 | 30Â min | HepG2 | ~900Â pmol/mg protein | Boulton et al. (1999)a |